{"id":552,"date":"2025-08-15T06:55:28","date_gmt":"2025-08-15T06:55:28","guid":{"rendered":"https:\/\/lwfzyzmd.com\/product\/%e5%8f%b8%e6%9b%bf%e6%88%8a%e9%86%87-%e7%94%a8%e4%ba%8e%e6%b2%bb%e7%96%976%e4%b8%aa%e6%9c%88%e5%8f%8a%e4%bb%a5%e4%b8%8a%e4%b8%94%e4%bd%93%e9%87%8d-7-kg%e7%9a%84%e6%9c%8d%e7%94%a8%e6%b0%af%e5%b7%b4\/"},"modified":"2026-09-23T00:37:38","modified_gmt":"2026-09-22T17:37:38","slug":"%e5%8f%b8%e6%9b%bf%e6%88%8a%e9%86%87-%e7%94%a8%e4%ba%8e%e6%b2%bb%e7%96%976%e4%b8%aa%e6%9c%88%e5%8f%8a%e4%bb%a5%e4%b8%8a%e4%b8%94%e4%bd%93%e9%87%8d-7-kg%e7%9a%84%e6%9c%8d%e7%94%a8%e6%b0%af%e5%b7%b4","status":"publish","type":"product","link":"https:\/\/laopharmacy.la\/th\/product\/%e5%8f%b8%e6%9b%bf%e6%88%8a%e9%86%87-%e7%94%a8%e4%ba%8e%e6%b2%bb%e7%96%976%e4%b8%aa%e6%9c%88%e5%8f%8a%e4%bb%a5%e4%b8%8a%e4%b8%94%e4%bd%93%e9%87%8d-7-kg%e7%9a%84%e6%9c%8d%e7%94%a8%e6%b0%af%e5%b7%b4\/","title":{"rendered":"Lucius LuciStir Stiripentol 250mg"},"content":{"rendered":"<p><strong>\u53f8\u66ff\u620a\u9187<\/strong><strong>\u8bf4\u660e\u4e66<\/strong><\/p>\n<p>\u5546\u54c1\u540d\u79f0\uff1aLuciStir<\/p>\n<p>\u751f\u4ea7\u5546\uff1a\u5362\u4fee\u65af\u5236\u836f\u00a0Lucius<\/p>\n<p>\u4e2d\u6587\u540d\u79f0\uff1a\u53f8\u66ff\u620a\u9187<\/p>\n<p>\u82f1\u6587\u540d\u79f0\uff1a\u00a0Stiripentol<\/p>\n<p>\u836f\u54c1\u6279\u51c6\u6587\u53f7\uff1a12\u00a0L 1053\/23<\/p>\n<p>&nbsp;<\/p>\n<p>&nbsp;<\/p>\n<p><strong>\u3010\u6982\u62ec\u3011<\/strong><\/p>\n<p>\u7528\u4e8e\u6cbb\u75976\u4e2a\u6708\u53ca\u4ee5\u4e0a\u4e14\u4f53\u91cd\u22657 kg\u7684\u670d\u7528\u6c2f\u5df4\u5360\u60a3\u8005\u7684 Dravet \u7efc\u5408\u5f81 (DS) \u76f8\u5173\u766b\u75eb\u53d1\u4f5c\u3002<\/p>\n<p>&nbsp;<\/p>\n<p><strong>\u3010\u9002\u5e94\u75c7\u3011<\/strong><\/p>\n<p>\u7528\u4e8e\u6cbb\u75976\u4e2a\u6708\u53ca\u4ee5\u4e0a\u4e14\u4f53\u91cd\u22657 kg\u7684\u670d\u7528\u6c2f\u5df4\u5360\u60a3\u8005\u7684 Dravet \u7efc\u5408\u5f81 (DS) \u76f8\u5173\u766b\u75eb\u53d1\u4f5c\u3002\u5c1a\u65e0\u4e34\u5e8a\u6570\u636e\u652f\u6301\u4f7f\u7528 \u53f8\u66ff\u620a\u9187\u4f5c\u4e3a\u5355\u836f\u6cbb\u7597 Dravet \u7efc\u5408\u5f81\u3002<\/p>\n<p>&nbsp;<\/p>\n<p><strong>\u3010\u89c4\u683c\u3011\u00a0\u00a0<\/strong><\/p>\n<p>250mg\/\u7247\uff0c60\u7247\/\u74f6<\/p>\n<p>&nbsp;<\/p>\n<p><strong>\u3010\u7528\u6cd5\u7528\u91cf\u3011<\/strong><\/p>\n<p>1\u3001\u63a8\u8350\u53e3\u670d\u5242\u91cf\u4e3a 50 mg\/kg\/\u5929\uff0c\u52062\u62163\u6b21\u7ed9\u836f\uff08\u537316.67 mg\/kg\u6bcf\u65e53\u6b21\u6216 25 mg\/kg \u6bcf\u65e52\u6b21\uff09\uff0c\u5177\u4f53\u53d6\u51b3\u4e8e\u60a3\u8005\u7684\u5e74\u9f84\u548c\u4f53\u91cd\u3002<\/p>\n<p>2\u3001\u5982\u679c\u7ed9\u5b9a\u53ef\u7528\u89c4\u683c\u65e0\u6cd5\u8fbe\u5230\u786e\u5207\u5242\u91cf\uff0c\u5219\u56db\u820d\u4e94\u5165\u81f3\u6700\u63a5\u8fd1\u7684\u53ef\u80fd\u5242\u91cf\u3002<\/p>\n<p>3\u3001\u6700\u5927\u63a8\u8350\u603b\u5242\u91cf\u4e3a3,000 mg\/\u5929\u3002<\/p>\n<p>&nbsp;<\/p>\n<p><strong>\u3010\u00a0\u4e0d\u826f\u53cd\u5e94\u3011<\/strong><\/p>\n<p><strong>\u00a0<\/strong>\u6700\u5e38\u89c1\u7684\u4e0d\u826f\u53cd\u5e94\uff08\u81f3\u5c1110%\u7684\u00a0LuciStir-\u6cbb\u7597\u60a3\u8005\u53d1\u751f\u4e14\u6bd4\u5b89\u6170\u5242\u7ec4\u66f4\u5e38\u89c1\uff09\u5305\u62ec\uff1a<\/p>\n<p>1\u3001\u55dc\u7761 (67%)\u3001\u98df\u6b32\u4e0b\u964d (45%)\u3001\u6fc0\u8d8a (27%)\u3001<\/p>\n<p>2\u3001\u5171\u6d4e\u5931\u8c03 (27%)\u3001\u4f53\u91cd\u4e0b\u964d (27%)\u3001\u5f20\u529b\u51cf\u9000 (24%)\u3001<\/p>\n<p>3\u3001\u6076\u5fc3 (15%)\u3001\u9707\u98a4(15%)\u3001\u6784\u97f3\u969c\u788d (12%) \u548c\u5931\u7720 (12%)<\/p>\n<p><strong>\u00a0<\/strong><\/p>\n<p><strong>\u3010<\/strong><strong>\u6ce8\u610f\u4e8b\u9879<\/strong><strong>\u3011<\/strong><\/p>\n<p>1\u3001\u55dc\u7761<\/p>\n<p>LuciStir\u00a0\u53ef\u5f15\u8d77\u55dc\u7761\u3002\u5728 Dravet \u7efc\u5408\u5f81\u60a3\u8005\u7684\u5bf9\u7167\u7814\u7a76\u4e2d\uff0cLuciStir-\u6cbb\u7597\u7ec4\u60a3\u8005\u7684\u55dc\u7761\u53d1\u751f\u7387\u4e3a67%\uff0c\u76f8\u6bd4\u4e4b\u4e0b\uff0c\u5b89\u6170\u5242\u7ec4\u60a3\u8005\u7684\u53d1\u751f\u7387\u4e3a23%\u3002\u4e24\u7ec4\u4e2d\u7684\u6240\u6709\u60a3\u8005\u5747\u5408\u5e76\u4f7f\u7528\u6c2f\u5df4\u5360\uff0c\u5df2\u77e5\u6c2f\u5df4\u5360\u4e5f\u4f1a\u5f15\u8d77\u55dc\u7761\u3002LuciStir\u4e0e\u6c2f\u5df4\u5360\u8054\u5408\u7ed9\u836f\u5bfc\u81f4\u6c2f\u5df4\u5360\u53ca\u5176\u6d3b\u6027\u4ee3\u8c22\u7269\u6c34\u5e73\u5347\u9ad8 [\u89c1\u836f\u7269\u76f8\u4e92\u4f5c\u7528 (7.1)]\u3002\u5176\u4ed6\u4e2d\u67a2\u795e\u7ecf\u7cfb\u7edf\u6291\u5236\u5242\uff08\u5305\u62ec\u9152\u7cbe\uff09\u53ef\u589e\u5f3a\u00a0LuciStir\u00a0\u7684\u55dc\u7761\u4f5c\u7528\u3002<\/p>\n<p>\u5904\u65b9\u533b\u751f\u5e94\u76d1\u6d4b\u60a3\u8005\u662f\u5426\u51fa\u73b0\u55dc\u7761\u3002\u5982\u679c\u5728\u4e0e\u6c2f\u5df4\u5360\u540c\u65f6\u7ed9\u836f\u671f\u95f4\u53d1\u751f\u55dc\u7761\uff0c\u8003\u8651\u6c2f\u5df4\u5360\u521d\u59cb\u5242\u91cf\u51cf\u5c1125%\u3002\u5982\u679c\u55dc\u7761\u6301\u7eed\u5b58\u5728\uff0c\u5e94\u8003\u8651\u8fdb\u4e00\u6b65\u5c06\u6c2f\u5df4\u5360\u51cf\u5c1125%\uff0c\u5e76\u5e94\u8c03\u6574\u5176\u4ed6\u5177\u6709\u9547\u9759\u4f5c\u7528\u7684\u5408\u5e76\u6297\u60ca\u53a5\u836f\u7269\u7684\u5242\u91cf\u3002<\/p>\n<p>\u5904\u65b9\u533b\u5e08\u5e94\u63d0\u9192\u60a3\u8005\u4e0d\u8981\u4ece\u4e8b\u9700\u8981\u7cbe\u795e\u8b66\u89c9\u7684\u5371\u9669\u6d3b\u52a8\uff0c\u5982\u64cd\u4f5c\u5371\u9669\u673a\u68b0\u6216\u673a\u52a8\u8f66\uff0c\u76f4\u81f3\u00a0LuciStir\u00a0\u5bf9\u7cbe\u795e\u8b66\u89c9\u7684\u5f71\u54cd\u5df2\u77e5\u3002<\/p>\n<p>2\u3001\u98df\u6b32\u4e0b\u964d\u548c\u4f53\u91cd\u4e0b\u964d<\/p>\n<p>LuciStir\u00a0\u53ef\u5f15\u8d77\u98df\u6b32\u548c\u4f53\u91cd\u4e0b\u964d\u3002\u5728 Dravet \u7efc\u5408\u5f81\u60a3\u8005\u7684\u5bf9\u7167\u7814\u7a76\u4e2d\uff0cLuciStir-\u6cbb\u7597\u60a3\u8005\u4e2d\u98df\u6b32\u4e0b\u964d\u7684\u53d1\u751f\u7387\u4e3a46%\uff0c\u76f8\u6bd4\u4e4b\u4e0b\uff0c\u5b89\u6170\u5242\u7ec4\u60a3\u8005\u4e3a10%\u3002LuciStir-\u6cbb\u7597\u7ec4\u60a3\u8005\u7684\u4f53\u91cd\u4e0b\u964d\u53d1\u751f\u7387\u4e3a27%\uff0c\u800c\u5b89\u6170\u5242\u7ec4\u60a3\u8005\u4e3a6%\u3002\u63a5\u53d7\u00a0LuciStir-\u6cbb\u7597\u7684\u60a3\u8005\u4e2d\u6076\u5fc3\u548c\u5455\u5410\u7684\u53d1\u751f\u7387\u4e5f\u66f4\u9ad8 [\u53c2\u89c1\u4e0d\u826f\u53cd\u5e94 (6.1)]\u3002\u9274\u4e8e\u8fd9\u4e9b\u4e0d\u826f\u53cd\u5e94\u7684\u9891\u7387\uff0c\u5e94\u4ed4\u7ec6\u76d1\u6d4b\u63a5\u53d7\u00a0LuciStir\u00a0\u6cbb\u7597\u7684\u513f\u79d1\u60a3\u8005\u7684\u751f\u957f\u3002\u5728\u67d0\u4e9b\u60c5\u51b5\u4e0b\uff0c\u5c06\u5408\u5e76\u4f7f\u7528\u7684\u4e19\u620a\u9178\u76d0\u5242\u91cf\u51cf\u5c1130%\/\u5468\u53ef\u51cf\u5c11\u98df\u6b32\u548c\u4f53\u91cd\u51cf\u8f7b\u3002<\/p>\n<p>3\u3001\u4e2d\u6027\u7c92\u7ec6\u80de\u51cf\u5c11\u75c7\u548c\u8840\u5c0f\u677f\u51cf\u5c11\u75c7<\/p>\n<p>LuciStir\u00a0\u53ef\u5f15\u8d77\u4e2d\u6027\u7c92\u7ec6\u80de\u8ba1\u6570\u663e\u8457\u4e0b\u964d\u3002\u5728 Dravet \u7efc\u5408\u5f81\u60a3\u8005\u7684\u5bf9\u7167\u7814\u7a76\u4e2d\uff0c31\u4f8b\u63a5\u53d7\u00a0LuciStir\u00a0\u6cbb\u7597\u7684\u60a3\u8005\u83b7\u5f97\u4e86\u57fa\u7ebf\u548c\u7814\u7a76\u7ed3\u675f\u4e2d\u6027\u7c92\u7ec6\u80de\u8ba1\u6570\u3002\u5728\u8fd9\u4e9b\u63a5\u53d7\u00a0LuciStir-\u6cbb\u7597\u7684\u60a3\u8005\u4e2d\uff0c\u670913%\u7684\u60a3\u8005\u5728\u8bd5\u9a8c\u671f\u95f4\u89c2\u5bdf\u5230\u4e2d\u6027\u7c92\u7ec6\u80de\u8ba1\u6570\u4ece\u57fa\u7ebf\u65f6\u6b63\u5e38\u964d\u4f4e\u81f3\u4f4e\u4e8e1500\u4e2a\u7ec6\u80de\/mm 3\uff0c\u4f46\u5728\u4efb\u4f55\u5b89\u6170\u5242\u6cbb\u7597\u7684\u60a3\u8005\u4e2d\u5747\u672a\u89c2\u5bdf\u5230\u3002<\/p>\n<p>LuciStir\u00a0\u53ef\u5f15\u8d77\u8840\u5c0f\u677f\u8ba1\u6570\u663e\u8457\u4e0b\u964d\u3002\u5728 Dravet \u7efc\u5408\u5f81\u60a3\u8005\u7684\u5bf9\u7167\u7814\u7a76\u4e2d\uff0c31\u4f8b\u63a5\u53d7\u00a0LuciStir\u00a0\u6cbb\u7597\u7684\u60a3\u8005\u5177\u6709\u57fa\u7ebf\u548c\u7814\u7a76\u7ed3\u675f\u8840\u5c0f\u677f\u8ba1\u6570\u3002\u572813%\u7684\u00a0LuciStir-\u6cbb\u7597\u60a3\u8005\u4e2d\u89c2\u5bdf\u5230\u8840\u5c0f\u677f\u8ba1\u6570\u4ece\u57fa\u7ebf\u65f6\u6b63\u5e38\u964d\u4f4e\u81f3\u8bd5\u9a8c\u671f\u95f4\u4f4e\u4e8e150,000\/\u00b5L\uff0c\u4f46\u5728\u4efb\u4f55\u5b89\u6170\u5242\u6cbb\u7597\u60a3\u8005\u4e2d\u5747\u672a\u89c2\u5bdf\u5230\u3002<\/p>\n<p>\u5e94\u5728\u5f00\u59cb\u00a0LuciStir\u00a0\u6cbb\u7597\u524d\u8fdb\u884c\u8840\u6db2\u5b66\u68c0\u67e5\uff0c\u7136\u540e\u6bcf6\u4e2a\u6708\u8fdb\u884c\u4e00\u6b21\u3002<\/p>\n<p>4\u3001\u6212\u65ad\u75c7\u72b6<\/p>\n<p>\u4e0e\u5927\u591a\u6570\u6297\u766b\u75eb\u836f\u7269\u4e00\u6837\uff0cLuciStir\u901a\u5e38\u5e94\u9010\u6e10\u505c\u836f\uff0c\u4ee5\u5c3d\u91cf\u51cf\u5c11\u766b\u75eb\u53d1\u4f5c\u9891\u7387\u589e\u52a0\u548c\u766b\u75eb\u6301\u7eed\u72b6\u6001\u7684\u98ce\u9669\u3002<\/p>\n<p>\u5728\u9700\u8981\u5feb\u901f\u505c\u7528\u00a0LuciStir\u00a0\u7684\u60c5\u51b5\u4e0b\uff08\u4f8b\u5982\uff0c\u5728\u4e25\u91cd\u4e0d\u826f\u53cd\u5e94\u7684\u60c5\u51b5\u4e0b\uff09\uff0c\u5efa\u8bae\u8fdb\u884c\u9002\u5f53\u76d1<\/p>\n<p>5\u3001\u82ef\u4e19\u916e\u5c3f\u75c7\u60a3\u8005\u7684\u98ce\u9669<\/p>\n<p>\u82ef\u4e19\u6c28\u9178\u5bf9\u82ef\u4e19\u916e\u5c3f\u75c7 (PKU) \u60a3\u8005\u53ef\u80fd\u6709\u5bb3\u3002LuciStir\u53e3\u670d\u6df7\u60ac\u5242\u542b\u6709\u82ef\u4e19\u6c28\u9178\uff0c\u4e00\u79cd\u963f\u65af\u5df4\u751c\u6210\u5206\u3002\u6bcf\u4e2a 250 mg \u5305\u88c5\u542b1.40 mg\u82ef\u4e19\u6c28\u9178\uff1b\u6bcf 500 mg \u5305\u88c5\u542b2.80 mg\u82ef\u4e19\u6c28\u9178\u3002\u5728\u4e3a PKU \u60a3\u8005\u5904\u65b9\u00a0LuciStir\u00a0\u53e3\u670d\u6df7\u60ac\u5242\u4e4b\u524d\uff0c\u8003\u8651\u6240\u6709\u6765\u6e90\u7684\u82ef\u4e19\u6c28\u9178\u6bcf\u65e5\u603b\u91cf\uff0c\u5305\u62ec\u00a0LuciStir\u00a0\u53e3\u670d\u6df7\u60ac\u5242\u3002<\/p>\n<p>LuciStir\u00a0\u80f6\u56ca\u4e0d\u542b\u82ef\u4e19\u6c28\u9178\u3002<\/p>\n<p>6\u3001\u81ea\u6740\u884c\u4e3a\u548c\u610f\u5ff5<\/p>\n<p>AED\uff08\u5305\u62ecLuciStir\uff09\u4f1a\u589e\u52a0\u670d\u7528\u8fd9\u4e9b\u836f\u7269\u6cbb\u7597\u4efb\u4f55\u9002\u5e94\u75c7\u7684\u60a3\u8005\u81ea\u6740\u60f3\u6cd5\u6216\u884c\u4e3a\u7684\u98ce\u9669\u3002\u63a5\u53d7\u4efb\u4f55 AED \u6cbb\u7597\u4efb\u4f55\u9002\u5e94\u75c7\u7684\u60a3\u8005\u5e94\u76d1\u6d4b\u6291\u90c1\u7684\u51fa\u73b0\u6216\u6076\u5316\u3001\u81ea\u6740\u60f3\u6cd5\u6216\u884c\u4e3a\u548c\/\u6216\u60c5\u7eea\u6216\u884c\u4e3a\u7684\u4efb\u4f55\u5f02\u5e38\u53d8\u5316\u3002<\/p>\n<p>\u4efb\u4f55\u8003\u8651\u5904\u65b9\u00a0LuciStir\u00a0\u6216\u4efb\u4f55\u5176\u4ed6 AED \u7684\u4eba\u5fc5\u987b\u5e73\u8861\u81ea\u6740\u60f3\u6cd5\u6216\u884c\u4e3a\u7684\u98ce\u9669\u4e0e\u672a\u6cbb\u7597\u75be\u75c5\u7684\u98ce\u9669\u3002\u766b\u75eb\u548c\u8bb8\u591a\u5176\u4ed6\u5904\u65b9 AED \u7684\u75be\u75c5\u672c\u8eab\u4e0e\u53d1\u75c5\u7387\u548c\u6b7b\u4ea1\u7387\u4ee5\u53ca\u81ea\u6740\u60f3\u6cd5\u548c\u884c\u4e3a\u98ce\u9669\u589e\u52a0\u76f8\u5173\u3002\u5982\u679c\u5728\u6cbb\u7597\u671f\u95f4\u51fa\u73b0\u81ea\u6740\u60f3\u6cd5\u548c\u884c\u4e3a\uff0c\u5904\u65b9\u533b\u751f\u9700\u8981\u8003\u8651\u4efb\u4f55\u7279\u5b9a\u60a3\u8005\u51fa\u73b0\u7684\u8fd9\u4e9b\u75c7\u72b6\u662f\u5426\u4e0e\u6b63\u5728\u6cbb\u7597\u7684\u75be\u75c5\u6709\u5173\u3002<\/p>\n<p>\u5e94\u544a\u77e5\u60a3\u8005\u3001\u5176\u62a4\u7406\u4eba\u5458\u548c\u5bb6\u5c5e AED \u4f1a\u589e\u52a0\u81ea\u6740\u60f3\u6cd5\u548c\u884c\u4e3a\u7684\u98ce\u9669\uff0c\u5e94\u544a\u77e5\u5176\u9700\u8981\u8b66\u60d5\u6291\u90c1\u4f53\u5f81\u548c\u75c7\u72b6\u7684\u51fa\u73b0\u6216\u6076\u5316\u3001\u60c5\u7eea\u6216\u884c\u4e3a\u7684\u4efb\u4f55\u5f02\u5e38\u53d8\u5316\u6216\u81ea\u6740\u60f3\u6cd5\u3001\u884c\u4e3a\u6216\u81ea\u6211\u4f24\u5bb3\u60f3\u6cd5\u7684\u51fa\u73b0\u3002\u5e94\u7acb\u5373\u5411\u533b\u7597\u4fdd\u5065\u63d0\u4f9b\u8005\u62a5\u544a\u5173\u6ce8\u7684\u884c\u4e3a\u3002<\/p>\n<p>&nbsp;<\/p>\n<p><strong>\u3010<\/strong><strong>\u7981\u5fcc\u75c7<\/strong><strong>\u3011<\/strong><\/p>\n<p>\u65e0<\/p>\n<p><strong>\u3010<\/strong><strong>\u836f\u7269\u76f8\u4e92\u4f5c\u7528<\/strong><strong>\u3011<\/strong><\/p>\n<p>1\u3001LuciStir\u00a0\u5bf9\u5176\u4ed6\u836f\u7269\u7684\u5f71\u54cd<\/p>\n<p>CYP1A2\u3001CYP2B6\u3001CYP3A4\u3001CYP2C8\u3001CYP2C19\u3001P-\u7cd6\u86cb\u767d (P-gp) \u548c\u4e73\u817a\u764c\u8010\u836f\u86cb\u767d (BCRP) \u5e95\u7269<\/p>\n<p>\u4f53\u5916\u6570\u636e\u663e\u793a\uff0c\u53f8\u66ff\u620a\u9187\u662fCYP1A2\u3001CYP2B6\u548c CYP3A4 \u7684\u6291\u5236\u5242\u548c\u8bf1\u5bfc\u5242\u3002\u7531\u4e8e\u6f5c\u5728\u7684\u836f\u7269\u76f8\u4e92\u4f5c\u7528\uff0c\u5f53\u4e0e\u00a0LuciStir\u00a0\u4f34\u968f\u7ed9\u836f\u65f6\uff0c\u5e94\u6839\u636e\u4e34\u5e8a\u60c5\u51b5\u8003\u8651\u8c03\u6574 CYP1A2 \u5e95\u7269\uff08\u5982\u8336\u78b1\u3001\u5496\u5561\u56e0\uff09\u3001CYP2B6\u5e95\u7269\uff08\u5982\u820d\u66f2\u6797\u3001\u585e\u66ff\u6d3e\uff09\u548c CYP3A4 \u5e95\u7269\uff08\u5982\u54aa\u8fbe\u5511\u4ed1\u3001\u4e09\u5511\u4ed1\u3001\u594e\u5c3c\u4e01\uff09\u7684\u5242\u91cf\u3002<\/p>\n<p>\u7531\u4e8e\u53ef\u80fd\u6291\u5236\u9176\/\u8f6c\u8fd0\u86cb\u767d\u6d3b\u6027\uff0c\u5982\u679c\u4e0e\u00a0LuciStir\u00a0\u4f34\u968f\u7ed9\u836f\u65f6\u53d1\u751f\u4e0d\u826f\u53cd\u5e94\uff0c\u5e94\u8003\u8651\u51cf\u5c11CYP2C8\u3001CYP2C19\u5e95\u7269\uff08\u5982\u5730\u897f\u6cee\u3001\u6c2f\u5421\u683c\u96f7\uff09\u3001P-gp\u5e95\u7269\uff08\u5982\u5361\u9a6c\u897f\u5e73\uff09\u548c BCRP \u5e95\u7269\uff08\u5982\u7532\u6c28\u8776\u5464\u3001\u54cc\u5511\u55ea\u3001\u683c\u5217\u672c\u8132\uff09\u7684\u5242\u91cf\u3002<\/p>\n<p>\u6c2f\u5df4\u5360<\/p>\n<p>LuciStir\uff08\u6291\u5236 CYP 3A4 \u548c2C19\uff09\u4e0e\u6c2f\u5df4\u5360\u5408\u7528\u5bfc\u81f4\u6c2f\u5df4\u5360\uff08CYP 3A4\u7684\u5e95\u7269\uff09\u548c\u53bb\u7532\u6c2f\u5df4\u5360\uff08\u6c2f\u5df4\u5360\u7684\u6d3b\u6027\u4ee3\u8c22\u7269\uff0cCYP2C19\u7684\u5e95\u7269\uff09\u7684\u8840\u6d46\u6d53\u5ea6\u5347\u9ad8\u3002<\/p>\n<p>\u8fd9\u53ef\u80fd\u4f1a\u589e\u52a0\u6c2f\u5df4\u5360\u76f8\u5173\u4e0d\u826f\u53cd\u5e94\u7684\u98ce\u9669\u3002\u5982\u679c\u4e0e\u00a0LuciStir\u00a0\u8054\u5408\u7ed9\u836f\u65f6\u53d1\u751f\u4e0d\u826f\u53cd\u5e94\uff0c\u8003\u8651\u51cf\u5c11\u6c2f\u5df4\u5360\u7684\u5242\u91cf [\u89c1\u8b66\u544a\u548c\u6ce8\u610f\u4e8b\u9879]\u3002<\/p>\n<p>2\u3001\u5176\u4ed6\u836f\u7269\u5bf9\u00a0LuciStir\u00a0\u7684\u5f71\u54cd<\/p>\n<p>\u5f53\u4e0eCYP1A2\u3001CYP3A4\u6216 CYP2C19 \u5f3a\u6548\u8bf1\u5bfc\u5242\uff08\u5982\u5229\u798f\u5e73\u3001\u82ef\u59a5\u82f1\u3001\u82ef\u5df4\u6bd4\u59a5\u548c\u5361\u9a6c\u897f\u5e73\uff09\u8054\u5408\u7ed9\u836f\u65f6\uff0c\u53ef\u80fd\u53d1\u751f\u5bfc\u81f4\u00a0LuciStir\u00a0\u6d53\u5ea6\u964d\u4f4e\u7684\u57fa\u4e8e\u8bf1\u5bfc\u7684\u76f8\u4e92\u4f5c\u7528\uff0c\u56e0\u4e3a\u8fd9\u4e9b\u9176\u5747\u53ef\u4ee3\u8c22\u53f8\u66ff\u620a\u9187\u3002<\/p>\n<p>\u5e94\u907f\u514d\u00a0LuciStir\u00a0\u4e0e\u5f3a\u8bf1\u5bfc\u5242\u5408\u5e76\u4f7f\u7528\uff0c\u6216\u8fdb\u884c\u5242\u91cf\u8c03\u6574\u3002<\/p>\n<p>3\u3001CNS \u6291\u5236\u5242\u548c\u9152\u7cbe<\/p>\n<p>LuciStir\u00a0\u4e0e\u5176\u4ed6 CNS \u6291\u5236\u5242\uff08\u5305\u62ec\u9152\u7cbe\uff09\u5408\u5e76\u4f7f\u7528\u53ef\u80fd\u589e\u52a0\u9547\u9759\u548c\u55dc\u7761\u7684\u98ce\u9669 [\u89c1\u8b66\u544a\u548c\u6ce8\u610f\u4e8b\u9879]\u3002<\/p>\n<p>&nbsp;<\/p>\n<p><strong>\u3010<\/strong><strong>\u836f\u7269\u8fc7\u91cf<\/strong><strong>\u3011<\/strong><\/p>\n<p>\u5c1a\u65e0\u5173\u4e8e\u4eba\u4f53\u7528\u836f\u8fc7\u91cf\u7684\u6570\u636e\u3002\u5728\u63a5\u53d7\u9ad8\u5242\u91cf\u53f8\u66ff\u620a\u9187 (600-1800 mg\/kg i.p.) \u7ed9\u836f\u7684\u5c0f\u9f20\u4e2d\uff09\u53ef\u89c1\u8fd0\u52a8\u6d3b\u52a8\u51cf\u5c11\uff0c\u547c\u5438\u51cf\u5f31\u3002<\/p>\n<p>\u836f\u7269\u8fc7\u91cf\u7684\u6cbb\u7597\u5e94\u662f\u652f\u6301\u6027\u7684\uff08\u5728\u91cd\u75c7\u76d1\u62a4\u5ba4\u91c7\u53d6\u5bf9\u75c7\u63aa\u65bd\uff09\u3002<\/p>\n","protected":false},"excerpt":{"rendered":"<p>\u53f8\u66ff\u620a\u9187\u8bf4\u660e\u4e66 \u5546\u54c1\u540d\u79f0\uff1aLuciStir \u751f\u4ea7\u5546\uff1a\u5362\u4fee\u65af\u5236\u836f\u00a0Lucius \u4e2d\u6587\u540d\u79f0\uff1a\u53f8\u66ff\u620a\u9187 \u82f1\u6587\u540d\u79f0\uff1a\u00a0 [&hellip;]<\/p>\n","protected":false},"featured_media":1182,"comment_status":"open","ping_status":"closed","template":"","meta":{"advanced_seo_description":"","jetpack_seo_html_title":"","jetpack_seo_noindex":false,"jetpack_seo_schema_type":""},"product_brand":[],"product_cat":[432],"product_tag":[],"class_list":["post-552","product","type-product","status-publish","has-post-thumbnail","product_cat-432","first","instock","sale","purchasable","product-type-simple"],"jetpack_sharing_enabled":true,"_links":{"self":[{"href":"https:\/\/laopharmacy.la\/th\/wp-json\/wp\/v2\/product\/552","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/laopharmacy.la\/th\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/laopharmacy.la\/th\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/laopharmacy.la\/th\/wp-json\/wp\/v2\/comments?post=552"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/laopharmacy.la\/th\/wp-json\/wp\/v2\/media\/1182"}],"wp:attachment":[{"href":"https:\/\/laopharmacy.la\/th\/wp-json\/wp\/v2\/media?parent=552"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/laopharmacy.la\/th\/wp-json\/wp\/v2\/product_brand?post=552"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/laopharmacy.la\/th\/wp-json\/wp\/v2\/product_cat?post=552"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/laopharmacy.la\/th\/wp-json\/wp\/v2\/product_tag?post=552"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}